平安! 发表于 2011-11-9 19:57
/ ~+ U: N v2 S, q' qPazopanib (100 mg/kg/day free base equivalent)
3 p, W! C* j2 b' v$ X% r" ?( C8 Q 这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。3 n |9 M, r; p+ h
搜索了一下,原料一大堆。# v; b5 I" W" n+ G$ s/ v+ C
8 N& O) C. G& M6 B% \% G对不起!100mg/kg是用于移植瘤的,我弄错了。
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以下是正版说明书的推荐用量。$ P" h. j" y5 U- U9 \
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--------------------- DOSAGE AND ADMINISTRATION ----------------
5 t5 `2 y* }+ t/ A* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1) * T+ v& v1 ?1 [+ p0 k4 R5 M
* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2) ( @- `* ^7 [5 |' H
---------------------DOSAGE FORMS AND STRENGTHS --------------' ]8 Z# _, I# k' o3 m
200 mg tablets. (3) ( Z3 R# v* n& I* } o, i
-------------------------------CONTRAINDICATIONS------------------------ |